論文リスト 当研究室に所属する前の川本先生の研究に関する論文

7) Ikumi Kuriwaki, Minoru Kameda, Kazuhiko, Iikubo, Hiroyuki Hisamichi, Yuichiro Kawamoto, Shigetoshi Kikuchi, Hiroyuki Moritomo, Tadashi Terasaka, Yoshinori Iwai, Atsushi Noda, Hiroshi Tomiyama, Aya Kikuchi, and Masaaki Hirano, Discovery of ASP5878: Synthesis and structure–activity relationships of pyrimidine derivatives as pan-FGFRs inhibitors with improved metabolic stability and suppressed hERG channel inhibitory activity, Bioorganic and Medicinal Chemistry, 2022, 59, 116657. 


6) Ikumi Kuriwaki, Minoru Kameda, Kazuhiko, Iikubo, Hiroyuki Hisamichi, Yuichiro Kawamoto, Shigetoshi Kikuchi, Hiroyuki Moritomo, Yutaka Kondoh, Tadashi Terasaka, Yasushi Amano, Yukihiro Tateishi, Yuka Echizen, Yoshinori Iwai, Atsushi Noda, Hiroshi Tomiyama, Taisuke Nakazawa, and Masaaki Hirano, Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency, Bioorganic and Medicinal Chemistry, 2021, 33, 116019.  


5) Ikumi Kuriwaki, Minoru Kameda, Hiroyuki Hisamichi, Shigetoshi Kikuchi, Kazuhiko, Iikubo, Yuichiro Kawamoto, Hiroyuki Moritomo, Yutaka Kondoh, Yasushi Amano, Yukihiro Tateishi, Yuka Echizen, Yoshinori Iwai, Atsushi Noda, Hiroshi Tomiyama, Tomoyuki Suzuki and Masaaki Hirano, Structure-based drug design of 1,3,5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2, Bioorganic and Medicinal Chemistry, 2020, 28, 115453.  


4) Yuichiro Kawamoto, Ryushi Seo, Nobuhito Murai, Hideki Hiyama, Hiromasa Oka, Identification of potent lysophosphatidic acid receptor 5 (LPA5) antagonists as potential analgesic agents, Bioorganic and Medicinal Chemistry, 2018, 26, 257-265.  


3) Yasuo Hirooka, Kazutada Ikeuchi, Yuichiro Kawamoto, Yusuke Akao, Takumi Furuta, Tomohiro Asakawa, Makoto Inai, Toshiyuki Wakimoto, Tohru Fukuyama, and Toshiyuki Kan, Enantioselective Synthesis of SB-203207, Organic Letters201416, 1646-1649.

2) Toshiyuki Kan, Yuichiro Kawamoto, Tomohiro Asakawa, Takumi Furuta, and Tohru Fukuyama, Synthetic Studies on Altemicidin: Stereocontrolled Construction of the Core Framework, Organic Letters200810, 169-171.

1) Toshiyuki Kan, Tohru Inoue, Yuichiro Kawamoto, Mitsuhiro Yonehara, and Tohru Fukuyama, A Novel Synthesis of Bicyclo[3.3.0]octane Ring System via a Desymmetric C-H Insertion Reaction, Synlett200610, 1583-1585.